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personal data approved: 2017. III. 09.
Personal data
György Keserű
name György Keserű
year of birth 1967
name of institution
Budapest University of Technology and Economics
Doctoral Council of the University (external member)
Semmelweis University, Budapest
Habilitation Committee of the University (external member)
doctoral school
BME George A. Olah Doctoral School of Chemistry and Chemical Technology (Core member)
(discipline) Habilitation Comittee and Doctoral Council (external member)
SE Doctoral School of Pharmaceutical Sciences (Announcer of research topic)
the share of work in the different doctoral schools. BME George A. Olah Doctoral School of Chemistry and Chemical Technology 60%
SE Doctoral School of Pharmaceutical Sciences 38%
BME GAODSCC (discipline) Habilitation Comittee and Doctoral Council (external member) 1%
BME Doctoral Council of the University (external member) 1%
accreditation statement submitted to: Budapest University of Technology and Economics
HAC accreditation
full compliance
(2015. I. 30.)
Contact details
E-mail address gy.keseruttk.mta.hu
phone number +36 1 382-6821
own web page
Academic title
scientific degree, title Ph.D.
year degree was obtained 1994
discipline to which degree belongs chemistry
institution granting the degree HAS
scientific degree, title DSc
year degree was obtained 2003
discipline to which degree belongs
institution granting the degree HAS
Employment
2013 - MTA Természettudományi Kutatóközpont (research institute, not university)
scientific consultant
Thesis topic supervisor
number of doctoral students supervised until now 9
number of students who fulfilled course requirements 6
students who obtained their degrees:
Dávid Bajusz PhD 2017  GAODSCC
Ákos Tarcsay PhD 2014  GAODSCC
Márton Vass PhD 2014  GAODSCC
(50%) Róbert Kiss PhD 2008  DSPS1-SE
Tímea Polgár PhD 2006  GAODSCC
György Tibor Balogh PhD 2003  GAODSCC
László Molnár PhD 2003  GAODSCC
(50%) Dóra Menyhárd PhD 1998  DSPS1-SE

students with degree granting in process:
Ádám Andor Kelemen PhD (2018/06)  GAODSCC
Dávid Bajusz PhD (2018/06)  
present PhD students:
Aaron Brian Keeley (PhD) (2020/08)  GAODSCC
Andrea Scarpino (PhD) (2020/08)  GAODSCC
László Petri (PhD) (2019/01)  GAODSCC
  Thesis topic proposals
Research
research area medicinal chemistry, drug design
research field in which current research is conducted chemistry
pharmaceutics
Publications
2016

Bajusz D, Ferenczy GG, Keseru GM: Discovery of Subtype Selective Janus Kinase (JAK) Inhibitors by Structure-Based Virtual Screening, JOURNAL OF CHEMICAL INFORMATION AND MODELING 56: (1) pp. 234-247.
type of document: Journal paper/Article
number of independent citations: 2
language: English
DOI 
2016

Kelemen AA, Kiss R, Ferenczy GG, Kovacs L, Flachner B, Lorincz Z, Keseru GM: Structure-Based Consensus Scoring Scheme for Selecting Class A Aminergic GPCR Fragments, JOURNAL OF CHEMICAL INFORMATION AND MODELING 56: (2) pp. 412-422.
type of document: Journal paper/Article
number of independent citations: 1
language: English
DOI 
2016

Keseru GM, Erlanson DA, Ferenczy GG, Hann MM, Murray CW, Pickett SD: Design Principles for Fragment Libraries: Maximizing the Value of Learnings from Pharma Fragment-Based Drug Discovery (FBDD) Programs for Use in Academia, JOURNAL OF MEDICINAL CHEMISTRY 59: (18) pp. 8189-8206.
type of document: Journal paper/Article
number of independent citations: 4
language: English
DOI 
2015

Tarcsay A, Keseru GM: Is there a link between selectivity and binding thermodynamics profiles?, DRUG DISCOVERY TODAY 20: (1) pp. 86-94.
type of document: Journal paper/Review paper
number of independent citations: 12
language: English
URL 
2015

Szőllősi Edit, Bobok Amrita, Kiss László, Vass Márton, Kurkó Dalma, Kolok Sándor, Visegrády András, Keserű György Miklós: Cell-based and virtual fragment screening for adrenergic a2C receptor agonists, BIOORGANIC & MEDICINAL CHEMISTRY 23: (14) pp. 3991-3999.
type of document: Journal paper/Article
number of independent citations: 3
language: Albanian
DOI 
2014

Hopkins Andrew L, Keserue Gyoergy M, Leeson Paul D, Rees David C, Reynolds Charles H: The role of ligand efficiency metrics in drug discovery, NATURE REVIEWS DRUG DISCOVERY 13: (2) pp. 105-121.
type of document: Journal paper/Article
number of independent citations: 190
language: English
URL 
2014

Vass M, Schmidt E, Horti F, Keseru GM: Virtual fragment screening on GPCRs: A case study on dopamine D3 and histamine H4 receptors, EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 77: (2) pp. 38-46.
type of document: Journal paper/Article
number of independent citations: 22
language: English
URL 
2012

Ákos Tarcsay, Kinga Nyíri, György M Keserű: The Impact of Lipophilic Efficiency on Compound Quality, JOURNAL OF MEDICINAL CHEMISTRY 55: (3) pp. 1252-1260.
type of document: Journal paper/Article
number of independent citations: 71
language: English
DOI 
2012

Michael M Hann, György M Keserű: Finding the sweet spot: the role of nature and nurture in medicinal chemistry, NATURE REVIEWS DRUG DISCOVERY 11: pp. 355-365.
type of document: Journal paper/Article
number of independent citations: 148
language: English
DOI 
2009

Keserü G M, Makara G M: The influence of lead discovery strategies on the properties of drug candidates, NATURE REVIEWS DRUG DISCOVERY 8: (3) pp. 203-212.
type of document: Journal paper/Article
number of independent citations: 273
language: English
DOI 
Number of independent citations to these publications:726 
Scientometric data
list of publications and citations
number of scientific publications that meet accreditation criteria:
238
number of scientific publications:
255
monographs and professional books:
3
monographs/books in which chapters/sections were contributed:
12 
number of independent citations to scientific publications and creative works:
3232
further relevant information regarding accreditation (in Hungarian)
egyetemi magántanár (2004-től) a Budapesti Műszaki és Gazdaságtudományi Egyetem Vegyészmérnöki és Biomérnöki Karán Molekulatervezés illetve Molekulamodellezés tantárgyak oktatása a Budapesti Műszaki és Gazdaságtudományi Egyetemen 1993-től minden szemeszterben Gyógyszertervezés tantárgy oktatása Budapesti Műszaki és Gazdaságtudományi Egyetemen, az Eötvös Loránd Tudományegyetemen, a Debreceni Egyetemen és a Pécsi Egyetemen 2010-től (to be translated)

 
All rights reserved © 2007, Hungarian Doctoral Council. Doctoral Council registration number at commissioner for data protection: 02003/0001. Program version: 2.2358 ( 2017. X. 31. )